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Celastrol reverses palmitic acid (PA)-caused TLR4-MD2 activation-dependent insulin resistance via disrupting MD2-related cellular binding to PA

Xue Zhang , Ying Wang , Hui-Ya Ge , Yi-Jun Gu , Fan-Fan Cao , et al.
Journal of Cellular Physiology, 2018, 233 (10), pp.6814-6824. ⟨10.1002/jcp.26547⟩
Journal articles inserm-02402031v1

Celastrol improves the therapeutic efficacy of EGFR-TKIs for non-small-cell lung cancer by overcoming EGFR T790M drug resistance

Ying Wang , Qiuyun Liu , Haojie Chen , Jun You , Bin Peng , et al.
Anti-Cancer Drugs, 2018, 29 (8), pp.748-755. ⟨10.1097/CAD.0000000000000647⟩
Journal articles inserm-02402025v1
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HSP90 inhibitor, celastrol, arrests human monocytic leukemia cell U937 at G0/G1 in thiol-containing agents reversible way.

Bin Peng , Limin Xu , Fanfan Cao , Tingxuan Wei , Chunxin Yang , et al.
Molecular Cancer, 2010, 9 (1), pp.79. ⟨10.1186/1476-4598-9-79⟩
Journal articles inserm-00668221v1
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Celastrol Reverses Palmitic Acid-Induced Insulin Resistance in HepG2 Cells via Restoring the miR-223 and GLUT4 Pathway

Xue Zhang , Xiao-Cheng Xue , Ying Wang , Fan-Fan Cao , Jun You , et al.
Canadian Journal of Diabetes, 2019, 43 (3), pp.165-172. ⟨10.1016/j.jcjd.2018.07.002⟩
Journal articles inserm-02402019v1