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Beta-hydroxyphosphonate ribonucleoside analogues derived from 4-substituted-1,2,3-triazoles as IMP/GMP mimics: synthesis and biological evaluation

Tai Nguyen Van , Audrey Hospital , Corinne Lionne , Lars P. Jordheim , Charles Dumontet , et al.
Beilstein Journal of Organic Chemistry, 2016, 12, pp.1476--1486. ⟨10.3762/bjoc.12.144⟩
Journal articles hal-01812668v1
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Resistance to gemcitabine in a human follicular lymphoma cell line is due to partial deletion of the deoxycytidine kinase gene.

Carlos María Galmarini , Marilyn L. Clarke , Lars Jordheim , Cheryl L. Santos , Emeline Cros , et al.
BMC Pharmacology, 2004, 4, pp.8. ⟨10.1186/1471-2210-4-8⟩
Journal articles inserm-00112022v1

Polymeric nanocapsules as drug carriers for sustained anticancer activity of calcitriol in breast cancer cells

Sabrina Nicolas , Marie-Alexandrine Bolzinger , Lars Petter Jordheim , Yves Chevalier , Hatem Fessi , et al.
International Journal of Pharmaceutics, 2018, 550 (1-2), pp.170-179. ⟨10.1016/j.ijpharm.2018.08.022⟩
Journal articles hal-02139822v1
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Intracellular Cytidine Deaminase Regulates Gemcitabine Metabolism in Pancreatic Cancer Cell Lines

Tormod K Bjånes , Lars Petter Jordheim , Jan Schjøtt , Tina Kamceva , Emeline Cros-Perrial , et al.
Drug Metabolism and Disposition, 2019, 48 (3), pp.153 - 158. ⟨10.1124/dmd.119.089334⟩
Journal articles hal-04164121v1

Regulation of tumor infiltrated innate immune cells by adenosine

Regina Strakhova , Octavia Cadassou , Emeline Cros-Perrial , Lars Petter Jordheim
Purinergic Signalling, 2020, 16 (3), pp.289-295. ⟨10.1007/s11302-020-09701-6⟩
Journal articles hal-04164137v1
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The cytosolic 5’-nucleotidase cN-II lowers the adaptability to glucose deprivation in human breast cancer cells

Gabriel Bricard , Octavia Cadassou , Laure-Estelle Cassagnes , Emeline Cros-Perrial , Léa Payen-Gay , et al.
Journal articles hal-01611275v1
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Detecting differential allelic expression using high-resolution melting curve analysis: application to the breast cancer susceptibility gene CHEK2.

Tú Nguyen-Dumont , Lars Jordheim , Jocelyne Michelon , Nathalie Forey , Sandrine Mckay-Chopin , et al.
BMC Medical Genomics, 2011, 4 (1), pp.39. ⟨10.1186/1755-8794-4-39⟩
Journal articles inserm-00663661v1

Un tour d’horizon du développement de biomarqueurs pour les anticorps PD-1 et PD-L1 en cancérologie

Lisa Chaput , Lars Petter Jordheim
Therapies, 2021, 76 (6), pp.597-615. ⟨10.1016/j.therap.2021.06.005⟩
Journal articles hal-04165133v1
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Characterization of T‐DM1‐resistant breast cancer cells

Juliette Sauveur , Louise Conilh , Sabine Beaumel , Kamel Chettab , Lars Petter Jordheim , et al.
Pharmacology Research & Perspectives, 2020, 8 (4), pp.e00617. ⟨10.1002/prp2.617⟩
Journal articles hal-03810029v1
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Enriched PUFA environment of Leishmania infantum promastigotes promotes the accumulation of lipid mediators and favors parasite infectivity towards J774 murine macrophages

Marine Leroux , Hana Bouazizi-Ben Messaoud , Céline Luquain-Costaz , Lars Jordheim , Pauline Le Faouder , et al.
Lipids, 2023, 58 (2), pp.81-92. ⟨10.1002/lipd.12365⟩
Journal articles hal-04158694v1

Combretastatin A-4 sulfur-containing heterocyclic derivatives: Synthesis, antiproliferative activities and molecular docking studies

Abdelfattah Faouzi , Alexandre Arnaud , Alexandre Bancet , Caroline Barette , Jordane Preto , et al.
European Journal of Medicinal Chemistry, 2021, 215, pp.113275. ⟨10.1016/j.ejmech.2021.113275⟩
Journal articles hal-04165108v1
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Transcriptional and Metabolic Investigation in 5′-Nucleotidase Deficient Cancer Cell Lines

Octavia Cadassou , Prescillia Forey , Christelle Machon , Edoardo Petrotto , Kamel Chettab , et al.
Cells, 2021, 10 (11), pp.2918. ⟨10.3390/cells10112918⟩
Journal articles hal-03810114v1
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A Proposed Methodology to Deal with the Impact of In Vitro Cellular Matrix on the Analytical Performances of a Targeted Metabolomic LC-HRMS Method

Jérôme Guitton , Floriane Gavotto , Emeline Cros-Perrial , Lars Petter Jordheim , Christelle Machon
International Journal of Molecular Sciences, 2023, 24 (4), pp.3770. ⟨10.3390/ijms24043770⟩
Journal articles hal-04165175v1
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Adipocyte-conditioned medium induces resistance of breast cancer cells to lapatinib

A. Geneste , M. Duong , L. Molina , L. Conilh , S. Beaumel , et al.
BMC Pharmacology and Toxicology, 2020, 21 (1), pp.61. ⟨10.1186/s40360-020-00436-z⟩
Journal articles hal-03810208v1
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Cytotoxic and Antitumoral Activity of N-(9H-purin-6-yl) Benzamide Derivatives and Related Water-soluble Prodrugs

Emeline Cros-Perrial , Steve Saulnier , Muhammad Zawwad Raza , Rémi Charmelot , David Egron , et al.
Current Molecular Pharmacology, 2022, 15 (6), pp.883-894. ⟨10.2174/1874467214666211014164406⟩
Journal articles hal-03809743v1
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Identification of allosteric inhibitors of the ecto-5'-nucleotidase (CD73) targeting the dimer interface

Rahila Rahimova , Simon Fontanel , Corinne Lionne , Lars Peter Jordheim , Suzanne Peyrottes , et al.
PLoS Computational Biology, 2018, 14 (1), pp.e1005943. ⟨10.1371/journal.pcbi.1005943⟩
Journal articles hal-01838257v1
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Cytosolic 5′-Nucleotidase II Silencing in Lung Tumor Cells Regulates Metabolism through Activation of the p53/AMPK Signaling Pathway

Rossana Pesi , Simone Allegrini , Mercedes Garcia-Gil , Lucia Piazza , Roberta Moschini , et al.
International Journal of Molecular Sciences, 2021, 22 (13), pp.7004. ⟨10.3390/ijms22137004⟩
Journal articles hal-04165114v1
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Rationally designed hyaluronic acid-based nano-complexes for pentamidine delivery

Flavia Carton , Yves Chevalier , Letizia Nicoletti , Małgorzata Tarnowska , Barbara Stella , et al.
International Journal of Pharmaceutics, 2019, 568, pp.118526. ⟨10.1016/j.ijpharm.2019.118526⟩
Journal articles hal-02841561v1
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PARP Inhibitors and Proteins Interacting with SLX4

Lars Petter Jordheim
Journal articles hal-04164299v1
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Second‐Generation CD73 Inhibitors Based on a 4,6‐Biaryl‐2‐thiopyridine Scaffold

Rayane Ghoteimi , Abdennour Braka , Céline Rodriguez , Emeline Cros‐perrial , Valentin Duvauchelle , et al.
ChemMedChem, 2023, 18 (7), pp.e202200594. ⟨10.1002/cmdc.202200594⟩
Journal articles hal-04165181v1
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Cytosolic 5′-Nucleotidase II Is a Sensor of Energy Charge and Oxidative Stress: A Possible Function as Metabolic Regulator

Rossana Pesi , Simone Allegrini , Francesco Balestri , Mercedes Garcia-Gil , Federico Cividini , et al.
Cells, 2021, 10 (1), pp.182. ⟨10.3390/cells10010182⟩
Journal articles hal-04164184v1
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Structural Insights into the Inhibition of Cytosolic 5'-Nucleotidase II (cN-II) by Ribonucleoside 5'-Monophosphate Analogues

Franck Gallier , Perrine Lallemand , Maïa Meurillon , Lars P. Jordheim , Charles Dumontet , et al.
PLoS Computational Biology, 2011, 7 (12), pp.e1002295. ⟨10.1371/journal.pcbi.1002295⟩
Journal articles hal-00675257v1