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authFullName_s : Philippe Delagrange
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Update on Melatonin Receptors. IUPHAR Review.

Ralf Jockers , Philippe Delagrange , Margarita L Dubocovich , Regina P Markus , Nicolas Renault , et al.
British Journal of Pharmacology, 2016, ⟨10.1002/BPH.13536⟩
Journal articles inserm-01335656v1
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Quinazoline and phthalazine derivatives as novel melatonin receptor ligands analogues of agomelatine

Raphaël Bolteau , Florian Descamps , Mohamed Ettaoussi , Daniel H. Caignard , Philippe Delagrange , et al.
European Journal of Medicinal Chemistry, 2020, 189, pp.112078. ⟨10.1016/j.ejmech.2020.112078⟩
Journal articles hal-03489716v1
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Synthesis and pharmacological evaluation of dual ligands for melatonin (MT1/MT2) and serotonin 5-HT2C receptor subtypes (II)

Mohamed Ettaoussi , Basile Peres , A Errazani , J.A. Boutin , Daniel-Henri Caignard , et al.
European Journal of Medicinal Chemistry, 2015, 90, pp.822-833. ⟨10.1016/j.ejmech.2014.12.021⟩
Journal articles hal-02060835v1
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Protein interactome mining defines melatonin MT 1 receptors as integral component of presynaptic protein complexes of neurons

Abla Benleulmi-Chaachoua , Lina Chen , Kate Sokolina , Victoria Wong , Igor Jurisica , et al.
Journal of Pineal Research, 2015, ⟨10.1111/jpi.12294⟩
Journal articles istex inserm-01244306v1
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A Generic Approach for the Purification of Signaling Complexes That Specifically Interact with the Carboxyl-terminal Domain of G Protein-coupled Receptors

Pascal Maurice , Avais M Daulat , Cédric Broussard , Julien Mozo , Guilhem Clary , et al.
Molecular and Cellular Proteomics, 2008, 7 (8), pp.1556-69. ⟨10.1074/mcp.M700435-MCP200⟩
Journal articles hal-02348044v1

Negative regulation of melatonin secretion by melatonin receptors in ovine pinealocytes

Julie Lépinay , Catherine Taragnat , Jean-Philippe Dubois , Didier Chesneau , Ralf Jockers , et al.
PLoS ONE, 2021, 16 (7), pp.1-20. ⟨10.1371/journal.pone.0255249⟩
Journal articles hal-03466812v1

Detection of the human GPR50 orphan seven transmembrane protein by polyclonal antibodies mapping different epitopes

Hassina Ould Hamouda , Patty Chen , Angélique Levoye , Nejla Sözer-Topçular , Avais M Daulat , et al.
Journal of Pineal Research, 2007, 43 (1), pp.10-15. ⟨10.1111/j.1600-079X.2007.00437.x⟩
Journal articles istex hal-02348068v1
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The orphan GPR50 receptor promotes constitutive TGFβ receptor signaling and protects against cancer development

Stefanie Wojciech , Raise Ahmad , Zakia Belaid-Choucair , Anne-Sophie Journé , Sarah Gallet , et al.
Nature Communications, 2018, 9 (1), pp.1216. ⟨10.1038/s41467-018-03609-x⟩
Journal articles inserm-04021787v1
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Impaired α-tubulin re-tyrosination leads to synaptic dysfunction and is a feature of Alzheimer’s disease

Leticia Peris , Xiaoyi Qu , Jean-Marc Soleilhac , Julie Parato , Fabien Lanté , et al.
Preprints, Working Papers, ... hal-03432440v1
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Melatonergic ligands: Design, synthesis and pharmacological evaluation of novel series of naphthofuranic derivatives

Elodie Landagaray , Mohamed Ettaoussi , Romain Duroux , J.A. Boutin , Daniel-Henri Caignard , et al.
European Journal of Medicinal Chemistry, 2016, 109, pp.360-370. ⟨10.1016/j.ejmech.2015.12.047⟩
Journal articles hal-02060776v1
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Purification and Identification of G Protein- coupled Receptor Protein Complexes under Native Conditions

Avais M Daulat , Pascal Maurice , Carine Froment , Jean-Luc Guillaume , Cedric Broussard , et al.
Molecular and Cellular Proteomics, 2007
Journal articles hal-02348074v1