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Genome-wide studies of nuclear receptors in cell fate decisions.
Marco-Antonio Mendoza-Parra
,
Hinrich Gronemeyer
Journal articles
inserm-00854329v1
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Highly potent naphthofuran-based retinoic acid receptor agonists.
Efrén Pérez Santín
,
Harshal Khanwalkar
,
Johannes J. Voegel
,
Pascal Collette
,
Pascale Mauvais
,
et al.
Journal articles
inserm-00384552v1
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Growth factor-antagonized rexinoid apoptosis involves permissive PPARgamma/RXR heterodimers to activate the intrinsic death pathway by NO.
Pattabhiraman Shankaranarayanan
,
Aurélie Rossin
,
Harshal Khanwalkar
,
Susana Alvarez
,
Rosana Alvarez
,
et al.
Journal articles
inserm-00420821v1
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TRAIL: at the center of drugable anti-tumor pathways
Nicole Clarke
,
Angela Nebbioso
,
Lucia Altucci
,
Hinrich Gronemeyer
Journal articles
hal-04142402v1
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Retinoid receptor subtype-selective modulators through synthetic modifications of RARgamma agonists.
Susana Alvarez
,
Rosana Alvarez
,
Harshal Khanwalkar
,
Pierre Germain
,
Géraldine Lemaire
,
et al.
Journal articles
istex
inserm-00420402v1
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Synthesis and pharmacological characterization of Disila-AM80 (Disila-tamibarotene) and Disila-AM580, silicon analogues of the RARalpha-selective retinoid agonists AM80 (Tamibarotene) and AM580.
Reinhold Tacke
,
Volker Müller
,
Matthias W. Büttner
,
W Peter Lippert
,
Rüdiger Bertermann
,
et al.
Journal articles
istex
inserm-00438709v1
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An Unexpected Mode Of Binding Defines BMS948 as A Full Retinoic Acid Receptor β (RARβ, NR1B2) Selective Agonist
Eswarkumar Nadendla
,
Catherine Teyssier
,
Vanessa Delfosse
,
Valérie Vivat
,
Gunasekaran Krishnasamy
,
et al.
Journal articles
hal-02273910v1
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Decryption of the retinoid death code in leukemia
Lucia Altucci
,
Hinrich Gronemeyer
Journal articles
istex
hal-04130437v1
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Fingering modulators of retinoic acid signaling identifies new prognostic marker for neuroblastoma.
Hinrich Gronemeyer
,
Arthur Zelent
Journal articles
inserm-00384302v1
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Retinoic acid protects human breast cancer cells against etoposide-induced apoptosis by NF-kappaB-dependent but cIAP2-independent mechanisms.
Ana Jiménez-Lara
,
Ana Aranda
,
Hinrich Gronemeyer
Journal articles
inserm-00668473v1
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Dual role of DR5 in death and survival signaling leads to TRAIL resistance in cancer cells
Yelyzaveta Shlyakhtina
,
Valeria Pavet-Portal
,
Hinrich Gronemeyer
Journal articles
hal-03677786v1
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Cloning of a mouse glucocorticoid modulatory element binding protein, a new member of the KDWK family
Ana M. Jimenez-Lara
,
Matthias J. S. Heine
,
Hinrich Gronemeyer
Journal articles
hal-04094343v1
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Guidelines for the use and interpretation of assays for monitoring cell death in higher eukaryotes.
Lorenzo Galluzzi
,
Stuart A. Aaronson
,
John Abrams
,
Emad S Alnemri
,
David W. Andrews
,
et al.
Journal articles
inserm-00420382v1
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Leukemia: beneficial actions of retinoids and rexinoids
Lucia Altucci
,
Emmanuelle Wilhelm
,
Hinrich Gronemeyer
Journal articles
istex
hal-04130441v1
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9-cis-retinoic acid analogues with bulky hydrophobic rings: new RXR-selective agonists
Rosana Alvarez
,
M. Jesús Vega
,
Sabrina Kammerer
,
Aurélie Rossin
,
Pierre Germain
,
et al.
Journal articles
istex
hal-04122966v1
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The coactivator TIF2 contains three nuclear receptor-binding motifs and mediates transactivation through CBP binding-dependent and -independent pathways
Johannes J. Voegel
,
Matthias J. Heine
,
Marc Tini
,
Valérie Vivat
,
Pierre Chambon
,
et al.
Journal articles
hal-04057107v1
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The function of TIF2/GRIP1 in mouse reproduction is distinct from those of SRC-1 and p/CIP
Martine Gehin
,
Manuel Mark
,
Christine Dennefeld
,
Andrée Dierich
,
Hinrich Gronemeyer
,
et al.
Journal articles
hal-04145149v1
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Conformational adaptation of agonists to the human nuclear receptor RAR gamma
Bruno P. Klaholz
,
Jean-Paul Renaud
,
André Mitschler
,
C. Zusi
,
Pierre Chambon
,
et al.
Journal articles
istex
hal-04017111v1
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Epimetheus - a multi-profile normalizer for epigenomic sequencing data
Mohamed Ashick Mohamed Saleem
,
Marco Antonio Mendoza Parra
,
Pierre Cholley
,
Matthias Blum
,
Hinrich Gronemeyer
Journal articles
hal-03677828v1
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Differential action on coregulator interaction defines inverse retinoid agonists and neutral antagonists.
Pierre Germain
,
Claudine Gaudon
,
Vivian Pogenberg
,
Sarah Sanglier
,
Alain van Dorsselaer
,
et al.
Journal articles
inserm-00420381v1
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Inference from RNA interference: Suggestions to our authors
Hinrich Gronemeyer
Journal articles
hal-03665614v1
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C3 halogen and c8'' substituents on stilbene arotinoids modulate retinoic Acid receptor subtype function.
Susana Alvarez
,
Harshal Khanwalkar
,
Rosana Alvarez
,
Cathie Erb
,
Claudio Martínez
,
et al.
Journal articles
inserm-00438635v1
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The KDM5 family is required for activation of pro-proliferative cell cycle genes during adipocyte differentiation
Ann-Sofie Brier
,
Anne Loft
,
Jesper Madsen
,
Thomas Rosengren
,
Ronni Nielsen
,
et al.
Journal articles
hal-03677803v1
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Reconstruction of gene regulatory networks reveals chromatin remodelers and key transcription factors in tumorigenesis
Valeriya Malysheva
,
Marco Antonio Mendoza Parra
,
Mohamed Ashick Mohamed Saleem
,
Hinrich Gronemeyer
Journal articles
hal-03686927v1
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Versatile copurification procedure for rapid isolation of homogeneous RAR-RXR heterodimers
Jaya Iyer
,
Dominique Bonnier
,
Florence Granger
,
Carole Peluso-Iltis
,
Virginie Andry
,
et al.
Journal articles
istex
hal-04057119v1
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Allosteric effects govern nuclear receptor action: DNA appears as a player.
Hinrich Gronemeyer
,
William Bourguet
Journal articles
inserm-00420377v1
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Patient-matched analysis identifies deregulated networks in prostate cancer to guide personalized therapeutic intervention
Akinchan Kumar
,
Yasenya Kasikci
,
Alaa Badredine
,
Karim Azzag
,
Marie L Quintyn Ranty
,
et al.
American Journal of Cancer Research, 2021, 11 (11), pp.5299-5318. ⟨10.1101/695999⟩
Journal articles
hal-03473404v1
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The nuclear receptor ligand-binding domain: structure and function
Dino Moras
,
Hinrich Gronemeyer
Journal articles
istex
hal-04057134v1
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Silicon analogues of the RXR-selective retinoid agonist SR11237 (BMS649): chemistry and biology.
W Peter Lippert
,
Christian Burschka
,
Kathrin Götz
,
Martin Kaupp
,
Diana Ivanova
,
et al.
Journal articles
inserm-00420365v1
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Selective class II HDAC inhibitors impair myogenesis by modulating the stability and activity of HDAC-MEF2 complexes.
Angela Nebbioso
,
Fabio Manzo
,
Marco Miceli
,
Mariarosaria Conte
,
Lucrezia Manente
,
et al.
Journal articles
inserm-00420167v1
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