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Design of a disulfide-less, pharmacologically inert, and chemically competent analog of maurocalcine for the efficient transport of impermeant compounds into cells.
Narendra Ram
,
Norbert Weiss
,
Isabelle Texier-Nogues
,
Sonia Aroui
,
Nicolas Andreotti
,
et al.
Journal articles
inserm-00355685v1
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Pharmacological profiling of Orthochirus scrobiculosus toxin 1 analogs with a trimmed N-terminal domain.
Stéphanie Mouhat
,
Georgeta Teodorescu
,
Daniel Homerick
,
Violeta Visan
,
Heike Wulff
,
et al.
Journal articles
inserm-00381703v1
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Increasing the molecular contacts between maurotoxin and Kv1.2 channel augments ligand affinity.
Sarrah M'Barek
,
Benjamin Chagot
,
Nicolas Andreotti
,
Violeta Visan
,
Pascal Mansuelle
,
et al.
Journal articles
istex
inserm-00381749v1
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D-Maurocalcine, a pharmacologically inert efficient cell-penetrating peptide analogue.
Cathy Poillot
,
Kaouthar Dridi
,
Hicham Bichraoui
,
Julien Pêcher
,
Sébastien Alphonse
,
et al.
Journal articles
inserm-00587800v1
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The impact of the fourth disulfide bridge in scorpion toxins of the alpha-KTx6 subfamily.
Louis Carrega
,
Amor Mosbah
,
Gilles Ferrat
,
Christine Beeton
,
Nicolas Andreotti
,
et al.
Journal articles
istex
inserm-00394177v1
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Critical amino acid residues of maurocalcine involved in pharmacology, lipid interaction and cell penetration.
Kamel Mabrouk
,
Narendra Ram
,
Sylvie Boisseau
,
Flavie Strappazzon
,
Amel Rehaim
,
et al.
Journal articles
inserm-00378029v1
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The interaction between the measles virus nucleoprotein and the Interferon Regulator Factor 3 relies on a specific cellular environment
Matteo Colombo
,
Jean-Marie Bourhis
,
Célia Chamontin
,
Carine Soriano
,
Stéphanie Villet
,
et al.
Journal articles
hal-02475099v1
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K+ channel types targeted by synthetic OSK1, a toxin from Orthochirus scrobiculosus scorpion venom.
Stéphanie Mouhat
,
Violeta Visan
,
S. Ananthakrishnan
,
Heike Wulff
,
Nicolas Andreotti
,
et al.
Journal articles
inserm-00381756v1
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