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Highly potent naphthofuran-based retinoic acid receptor agonists.
Efrén Pérez Santín
,
Harshal Khanwalkar
,
Johannes J. Voegel
,
Pascal Collette
,
Pascale Mauvais
,
et al.
Journal articles
inserm-00384552v1
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Growth factor-antagonized rexinoid apoptosis involves permissive PPARgamma/RXR heterodimers to activate the intrinsic death pathway by NO.
Pattabhiraman Shankaranarayanan
,
Aurélie Rossin
,
Harshal Khanwalkar
,
Susana Alvarez
,
Rosana Alvarez
,
et al.
Journal articles
inserm-00420821v1
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Retinoid receptor subtype-selective modulators through synthetic modifications of RARgamma agonists.
Susana Alvarez
,
Rosana Alvarez
,
Harshal Khanwalkar
,
Pierre Germain
,
Géraldine Lemaire
,
et al.
Journal articles
istex
inserm-00420402v1
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Synthesis and pharmacological characterization of Disila-AM80 (Disila-tamibarotene) and Disila-AM580, silicon analogues of the RARalpha-selective retinoid agonists AM80 (Tamibarotene) and AM580.
Reinhold Tacke
,
Volker Müller
,
Matthias W. Büttner
,
W Peter Lippert
,
Rüdiger Bertermann
,
et al.
Journal articles
istex
inserm-00438709v1
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C3 halogen and c8'' substituents on stilbene arotinoids modulate retinoic Acid receptor subtype function.
Susana Alvarez
,
Harshal Khanwalkar
,
Rosana Alvarez
,
Cathie Erb
,
Claudio Martínez
,
et al.
Journal articles
inserm-00438635v1
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New retinoid chemotypes: 9-cis-retinoic acid analogs with hydrophobic rings derived from terpenes as selective RAR agonists.
Susana Alvarez
,
Yolanda Pazos-Randulfe
,
Harshal Khanwalkar
,
Pierre Germain
,
Rosana Alvarez
,
et al.
Journal articles
istex
inserm-00350716v1
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Pyrazine arotinoids with inverse agonist activities on the retinoid and rexinoid receptors.
José García
,
Harshal Khanwalkar
,
Raquel Pereira
,
Cathie Erb
,
Johannes J. Voegel
,
et al.
Journal articles
istex
inserm-00383337v1
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