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authFullName_s : Harshal Khanwalkar

Highly potent naphthofuran-based retinoic acid receptor agonists.

Efrén Pérez Santín , Harshal Khanwalkar , Johannes J. Voegel , Pascal Collette , Pascale Mauvais , et al.
ChemMedChem, 2009, 4 (5), pp.780-91. ⟨10.1002/cmdc.200900015⟩
Journal articles inserm-00384552v1

Growth factor-antagonized rexinoid apoptosis involves permissive PPARgamma/RXR heterodimers to activate the intrinsic death pathway by NO.

Pattabhiraman Shankaranarayanan , Aurélie Rossin , Harshal Khanwalkar , Susana Alvarez , Rosana Alvarez , et al.
Cancer Cell, 2009, 16 (3), pp.220-31. ⟨10.1016/j.ccr.2009.07.029⟩
Journal articles inserm-00420821v1

Retinoid receptor subtype-selective modulators through synthetic modifications of RARgamma agonists.

Susana Alvarez , Rosana Alvarez , Harshal Khanwalkar , Pierre Germain , Géraldine Lemaire , et al.
Bioorganic and Medicinal Chemistry, 2009, 17 (13), pp.4345-59. ⟨10.1016/j.bmc.2009.05.035⟩
Journal articles istex inserm-00420402v1

Synthesis and pharmacological characterization of Disila-AM80 (Disila-tamibarotene) and Disila-AM580, silicon analogues of the RARalpha-selective retinoid agonists AM80 (Tamibarotene) and AM580.

Reinhold Tacke , Volker Müller , Matthias W. Büttner , W Peter Lippert , Rüdiger Bertermann , et al.
ChemMedChem, 2009, 4 (11), pp.1797-802. ⟨10.1002/cmdc.200900257⟩
Journal articles istex inserm-00438709v1

C3 halogen and c8'' substituents on stilbene arotinoids modulate retinoic Acid receptor subtype function.

Susana Alvarez , Harshal Khanwalkar , Rosana Alvarez , Cathie Erb , Claudio Martínez , et al.
ChemMedChem, 2009, 4 (10), pp.1630-40. ⟨10.1002/cmdc.200900214⟩
Journal articles inserm-00438635v1

New retinoid chemotypes: 9-cis-retinoic acid analogs with hydrophobic rings derived from terpenes as selective RAR agonists.

Susana Alvarez , Yolanda Pazos-Randulfe , Harshal Khanwalkar , Pierre Germain , Rosana Alvarez , et al.
Bioorganic and Medicinal Chemistry, 2008, 16 (22), pp.9719-28. ⟨10.1016/j.bmc.2008.09.069⟩
Journal articles istex inserm-00350716v1

Pyrazine arotinoids with inverse agonist activities on the retinoid and rexinoid receptors.

José García , Harshal Khanwalkar , Raquel Pereira , Cathie Erb , Johannes J. Voegel , et al.
ChemBioChem, 2009, 10 (7), pp.1252-9. ⟨10.1002/cbic.200900030⟩
Journal articles istex inserm-00383337v1